Manufacturer: MaxtremePack: 10mg 50 pillsChemical Substance: Tamoxifen citrate (Nolvadex)
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Maxi-Fen-10 belongs to the group of anti-estrogenic drugs. The action of Maxi-Fen-10 is justified by its ability to block estrogen receptors. Maxi-Fen-10 competes with estradiol for binding sites with cytoplasmic estrogen receptors in the tissues of the breast, which makes Maxi-Fen-10 an effective tool in the fight against gynecomastia. However, Maxi-Fen-10 can not be used on a course with nandrolons and trenbolons. Maxi-Fen-10 has a fairly extensive list of side effects, in some of them: vision impairment, nausea, vomiting. The drug is toxic to the liver.
Tamoxifen can be used on a course to prevent gynecomastia, and it is also used during PCT (Post-course therapy). The dosage of tamoxifen is selected individually, according to the results of hormonal analyzes, usually starts from 10 mg.
Tamoxifen is an antimetabolite (antiestrogen) that competitively binds to estrogen receptors in the cytoplasm of estrogen-dependent tumor cells. Together with them, it penetrates into the nucleus, where it blocks the interaction of estrogens with its receptors.
After oral administration, the drug is rapidly absorbed and maximum serum concentrations are reached within 4-7 hours.
Stable concentrations (approximately 300 ng / ml) are achieved after a four-week treatment with a daily intake of 40 mg. Tamoxifen binds well to serum albumin (> 99%). As a result of metabolism, in the process of hydroxylation, demethylation and conjugation, a number of metabolites are formed, having pharmacological profile similar to the initial chemical compound, thus contributing to the achievement of a therapeutic effect. The half-life is 7 days. Isolation occurs mainly through feces.
Maxi-Fen-10 is a powerful and one of the most popular anti-estrogen bodybuilders. It avoids such phenomena of feminization as gynecomastia, which often appear at the end of the steroid cycle, as well as the accumulation of fat and water in the thigh or chest area. As a result, at the end of the cycle, most of the anabolic steroids are flavored into the hormone of estrogen, causing the appearance of feminization syndromes. Maxi-Fen-10 has the ability to block the receptors of estrogen, preventing it from manifesting the action and causing these phenomena. Many bodybuilders take Nolvadex before the competition, as it not only prevents the emergence of gynecomastia, but also reduces the accumulation of fat and water, which helps bodybuilders find a dried body.